BDBM50538869 CHEMBL4643188

SMILES CCNC(=O)c1cnc2ccc(nc2c1N[C@H]1CC[C@H](CN(C)C)CC1)-c1ccnc(N)c1

InChI Key InChIKey=LDTWDTRUGHYMIA-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50538869   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Stanford University

Curated by ChEMBL

LigandBDBM50538869(CHEMBL4643188)Copy SMILESCopy InChI

Affinity DataEC50:  46nMAssay Description:Inhibition of human DYRK1A transfected in HEK293T cells co-transfected with Renilla plasmid, pGL3-NFAT and NFATc1 assessed as derepression of NFAT-de...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/12/2021
Entry Details Article
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