BDBM50544518 CHEMBL4643133

SMILES [H][C@@]12Cc3c(CN1C(=O)N(Cc1ccc(F)cc1)C2=O)[nH]c1ccccc31

InChI Key InChIKey=QNJROIINZRKOAI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50544518   

TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Salerno

Curated by ChEMBL

LigandBDBM50544518(CHEMBL4643133)Copy SMILESCopy InChI

Affinity DataIC50: 1.78E+4nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium flux preincubated for 60 mins followed b...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/13/2021
Entry Details Article
Copy BDB DOIPubMed
Copy reaction URL