BDBM50544519 CHEMBL4640958

SMILES [H][C@@]12Cc3c([nH]c4ccccc34)[C@@H](CC(C)C)N1C(=O)N(Cc1ccc(OC)cc1)C2=O

InChI Key InChIKey=IAZBBHYVQSVMAS-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50544519   

TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Salerno

Curated by ChEMBL

LigandBDBM50544519(CHEMBL4640958)Copy SMILESCopy InChI

Affinity DataIC50: 2.80E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium flux preincubated for 60 mins followed b...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/13/2021
Entry Details Article
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