BDBM50544529 CHEMBL4640675

SMILES [H][C@@]12Cc3c([nH]c4ccccc34)[C@H](N1C(=O)N(C2=O)c1cccc(c1)C(F)(F)F)c1ccc(F)cc1

InChI Key InChIKey=BKIVSJZNZNFDNY-JTHBVZDNSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50544529   

TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50544529(CHEMBL4640675)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium flux preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed