BDBM50544533 CHEMBL4635623

SMILES [H][C@]12Cc3c([nH]c4ccccc34)[C@@H](N1C(=O)N(C2=O)c1ccccc1F)c1ccc(F)cc1

InChI Key InChIKey=YTCVHZUGAOACSA-GGAORHGYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50544533   

TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50544533(CHEMBL4635623)
Affinity DataIC50:  5.10E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium flux preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed