BDBM50549173 CHEMBL4789088

SMILES COc1cc(OC)cc(c1)C(=O)c1cn(C)c2nc(Nc3ccccc3NC(=O)C=C)ccc12

InChI Key InChIKey=CTOGOKDZTMAQHM-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50549173   

TargetFibroblast growth factor receptor 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50549173(CHEMBL4789088)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human FGFR4 using poly (Glu, Tyr)4:1 as substrate incubated for 20 mins followed by [33P]-ATP addition and measured after 120 mins by r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50549173(CHEMBL4789088)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of N-terminal GST tagged FGFR4 (unknown origin) expressed in baculovirus infected sf21 insect cells incubated for 2 hrs by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed