BDBM50558234 CHEMBL4780536

SMILES COc1cc(N)c(Cl)cc1C(=O)CCC1CCN(CCNS(=O)(=O)c2ccc(N)c(Br)c2)CC1

InChI Key InChIKey=LGPOBVLZHCYRKV-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50558234   

Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-GR113808 from guinea pig brain 5HT4 receptor in presence of serotonin incubated for 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]+/-DOI from human recombinant 5-HT2C receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor expressed in HEK293 cells in presence of serotonin incubated for 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Normandie Universit£

Curated by ChEMBL
LigandPNGBDBM50558234(CHEMBL4780536)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]ketanserin human recombinant 5-HT2A receptor after 60 mins by scintillation counting analysis relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed