BDBM50559824 CHEMBL4783963

SMILES CCc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(F)c1

InChI Key InChIKey=GHWMVXHLEAWLMB-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50559824   

TargetN-formyl peptide receptor 2(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50559824(CHEMBL4783963)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at human FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetfMet-Leu-Phe receptor(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50559824(CHEMBL4783963)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human FPR1 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed