BDBM50561524 CHEMBL4791756

SMILES Fc1ccc(Br)cc1Nc1ncnc2cc3OCCOc3cc12

InChI Key InChIKey=LUDNOLWHKWSFBJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50561524   

TargetEpidermal growth factor receptor(Human)
University of California, Los Angeles

Curated by ChEMBL
LigandPNGBDBM50561524(CHEMBL4791756)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human recombinant EGFR expressed in baculovirus infected Sf9 insect cells using poly (Glu, Tyr) 4:1 peptide as substrate incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of California, Los Angeles

Curated by ChEMBL
LigandPNGBDBM50561524(CHEMBL4791756)
Affinity DataIC50: 11nMAssay Description:Inhibition of wild type EGFR in human U87 cells assessed as heparin/human EGF stimulated phosphorylation after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed