BDBM50563557 CHEMBL4790791

SMILES Cn1cc(cn1)-c1coc2ccc(nc12)-c1cn[nH]c1

InChI Key InChIKey=SDHAXXDYIZVWAZ-UHFFFAOYSA-N

Data  5 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50563557   

TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL

LigandBDBM50563557(CHEMBL4790791)Copy SMILESCopy InChI

Affinity DataIC50:  176nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL

LigandBDBM50563557(CHEMBL4790791)Copy SMILESCopy InChI

Affinity DataIC50:  45nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL

LigandBDBM50563557(CHEMBL4790791)Copy SMILESCopy InChI

Affinity DataIC50:  28nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL

LigandBDBM50563557(CHEMBL4790791)Copy SMILESCopy InChI

Affinity DataIC50:  235nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Masaryk University

Curated by ChEMBL

LigandBDBM50563557(CHEMBL4790791)Copy SMILESCopy InChI

Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of human full length recombinant DYRK2 using casein substrate by radiometric scintillation assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
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