BDBM50563557 CHEMBL4790791

SMILES Cn1cc(cn1)-c1coc2ccc(nc12)-c1cn[nH]c1

InChI Key InChIKey=SDHAXXDYIZVWAZ-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50563557   Sort by

TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563557(CHEMBL4790791)
Affinity DataIC50: 176nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563557(CHEMBL4790791)
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50563557(CHEMBL4790791)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human full length recombinant DYRK2 using casein substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563557(CHEMBL4790791)
Affinity DataIC50: 235nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563557(CHEMBL4790791)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed