BDBM50563573 CHEMBL4742723

SMILES CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)C(=O)Nc1ccccc1

InChI Key InChIKey=HUXZYRMNXVAVPZ-CHQNGUEUSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50563573   

TargetProteasome subunit beta type-8(Homo sapiens (Human))
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50563573(CHEMBL4742723)
Affinity DataIC50:  231nMAssay Description:Inhibition of 20S immunoproteasome beta 5 chymotrypsin-like activity in human H226 cell using Suc-LLVY-AMC as substrate for 10 mins by fluorescence b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed