BDBM50570949 CHEMBL4848921
SMILES CC(C)NC(=O)c1cc(cnc1N)-c1ccc(NC(=O)[C@@](C)(O)c2ccccc2)cc1C
InChI Key InChIKey=DZDRNVJHVMKPKJ-VWLOTQADSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50570949
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of eIF2alpha (unknown origin) assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Homo sapiens (Human))
Hibercell
Curated by ChEMBL
Hibercell
Curated by ChEMBL
Affinity DataIC50: 159nMAssay Description:Inhibition of human His-tagged PERK expressed in Escherichia coli assessed as eIF2alpha phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair