BDBM50579183 CHEMBL4854949

SMILES CS(=O)(=O)c1ccc(\C=C\C2CC(Nc3ccnc(c3)-c3cc(F)ccc3F)=CC=N2)cc1

InChI Key InChIKey=CRDUMPVQRUQRQG-QHHAFSJGSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50579183   

TargetTGF-beta receptor type-1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50579183(CHEMBL4854949)
Affinity DataIC50:  13nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed