BDBM50584992 CHEMBL5085734
SMILES CC(C)c1ccccc1-c1nc(NCc2ccccn2)c2n(C)ccc2n1
InChI Key InChIKey=XIEZMAUGHWKZDR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50584992
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 beta(Human)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: <2.51E+4nMAssay Description:Inhibition of PI5P4Kbeta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Human)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: <5.01E+4nMAssay Description:Inhibition of PI5P4Kalpha (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 alpha(Human)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PI5P4Kalpha (unknown origin) incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 gamma(Human)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKd: 68nMAssay Description:Binding affinity to PI5P4Kgamma (unknown origin) by KINOMEscan analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 beta(Human)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to PI5P4Kbeta (unknown origin) by KINOMEscan analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 5-phosphate 4-kinase type-2 gamma(Human)
University of Cambridge
Curated by ChEMBL
University of Cambridge
Curated by ChEMBL
Affinity DataIC50: 794nMAssay Description:Binding affinity to ePL-tagged wild type PI5P4Kgamma (unknown origin) expressed in HEK293 cells incubated for 60 mins by InCell pulse thermal stabili...More data for this Ligand-Target Pair