BDBM50596594 CHEMBL5182936

SMILES CCCn1c2CCNC(=O)c2cc1-c1ccncc1

InChI Key InChIKey=AUMWRYOMDFANOB-UHFFFAOYSA-N

Data  2 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50596594   

TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596594(CHEMBL5182936)
Affinity DataKi:  7nMAssay Description:Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596594(CHEMBL5182936)
Affinity DataKi:  60nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596594(CHEMBL5182936)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of NanoLuc-PKN2 (ser646-cys984)(unknown origin) expressed in HEK293 cells by cell-based NanoBRET target engagement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596594(CHEMBL5182936)
Affinity DataIC50:  120nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50596594(CHEMBL5182936)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed