BDBM50600507 CHEMBL5173510

SMILES NC(=O)c1cc2c(cccc2s1)-c1cc(N)c(s1)C(=O)NC1CC1

InChI Key InChIKey=IIGCQCAUAFMZHK-UHFFFAOYSA-N

Data  2 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50600507   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Ach£

Curated by ChEMBL

LigandBDBM50600507(CHEMBL5173510)Copy SMILESCopy InChI

Affinity DataKi:  90nMAssay Description:Inhibition of human DYRK1A incubated for 90 mins in presence of ATP by Z-LYTE based FRET assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Ach£

Curated by ChEMBL

LigandBDBM50600507(CHEMBL5173510)Copy SMILESCopy InChI

Affinity DataKi:  814nMAssay Description:Inhibition of human DYRK1B incubated for 130 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI
Copy reaction URL