BDBM50613665 CHEMBL5266721

SMILES Cc1ccc2nc(n(-c3ccc(cc3)C(=O)CN3C(=O)NC4(CCC(F)(F)CC4)C3=O)c2n1)C(F)(F)F

InChI Key InChIKey=FFWJTSZVLJKGAJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50613665   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50613665(CHEMBL5266721)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK293 cells assessed as reduction in menthol induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed