BDBM50613791 CHEMBL4092332

SMILES COc1ccc(cc1)-n1nc2c(c[nH]c3cc(Br)ccc23)c1=O

InChI Key InChIKey=CAJJWNTVLDPILI-UHFFFAOYSA-N

Data  9 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50613791   

TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  1nMAssay Description:Positive allosteric modulation of rat recombinant GABAA alpha6beta3gamma2 receptor expressed in Xenopus laevis oocytes assessed as increase in GABA-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  4nMAssay Description:Positive allosteric modulation of rat recombinant GABAA gamma2beta3alpha1-beta3alpha6 receptor expressed in Xenopus laevis oocytes assessed as increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  9nMAssay Description:Positive allosteric modulation of rat recombinant GABAA alpha6beta3alpha6-gamma2beta3 receptor expressed in Xenopus laevis oocytes assessed as increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  6.00E+3nMAssay Description:Positive allosteric modulation of rat recombinant GABAA alpha1beta3gamma2 receptor expressed in Xenopus laevis oocytes assessed as increase in GABA-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  7.00E+3nMAssay Description:Positive allosteric modulation of rat recombinant GABAA alpha6beta3alpha1-gamma2beta3 receptor expressed in Xenopus laevis oocytes assessed as increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  1.00E+4nMAssay Description:Positive allosteric modulation of rat recombinant GABAA alpha1beta3alpha1-gamma2beta3 receptor expressed in Xenopus laevis oocytes assessed as increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  1.10E+4nMAssay Description:Positive allosteric modulation of rat recombinant GABAA alpha6beta3gamma2 receptor expressed in Xenopus laevis oocytes assessed as increase in GABA-i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  2.40E+4nMAssay Description:Positive allosteric modulation of rat recombinant GABAA alpha6beta3alpha6-gamma2beta3 receptor expressed in Xenopus laevis oocytes assessed as increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50613791(CHEMBL4092332)
Affinity DataEC50:  3.60E+4nMAssay Description:Positive allosteric modulation of rat recombinant GABAA gamma2beta3alpha1-beta3alpha6 receptor expressed in Xenopus laevis oocytes assessed as increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed