BDBM50617733 CHEMBL5410996

SMILES CN(Cc1ccccc1)c1ncnc2[nH]c(nc12)-c1ccccc1

InChI Key InChIKey=PPPZFHSMUGRPLW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50617733   

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Norwegian University of Science and Technology (NTNU)

US Patent
LigandChemical structure of BindingDB Monomer ID 50617733BDBM50617733(CHEMBL5410996 | US20250353857, Compound TIA072)
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2026
Entry Details US Patent

TargetMacrophage colony-stimulating factor 1 receptor(Human)
Norwegian University of Science and Technology (NTNU)

US Patent
LigandChemical structure of BindingDB Monomer ID 50617733BDBM50617733(CHEMBL5410996 | US20250353857, Compound TIA072)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of CSF1R (unknown origin) using FRET-peptide as substrate incubated in presence of ATP by FRET based Z-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed