BDBM50621214 CHEMBL5410094

SMILES CC(=O)\C=C1/Sc2ccc(O)cc2N1Cc1cccc(C)c1

InChI Key InChIKey=PRCDPUXQFRMFMC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50621214   

TargetDual specificity protein kinase CLK1(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandPNGBDBM50621214(CHEMBL5410094)
Affinity DataIC50: 39nMAssay Description:Inhibition of human CLK1 using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of Mg/[gamma-33P]-ATP by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of Rouen Normandy

Curated by ChEMBL
LigandPNGBDBM50621214(CHEMBL5410094)
Affinity DataIC50: 429nMAssay Description:Inhibition of human DYRK1A using RRRFRPASPLRGPPK as substrate incubated for 40 mins in presence of Mg/[gamma-33P]-ATP by scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed