BDBM50622252 CHEMBL5423911

SMILES COc1cc(CNC(=O)CCCc2cccs2)ccc1O

InChI Key InChIKey=HCUVEUVIUAJXRB-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50622252   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Magna Gracia University

Curated by ChEMBL
LigandPNGBDBM50622252(CHEMBL5423911)
Affinity DataEC50:  870nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Magna Gracia University

Curated by ChEMBL
LigandPNGBDBM50622252(CHEMBL5423911)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as desensitization by measuring inhibition of capsaicin-induced int...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed