BDBM50622581 CHEMBL5402691

SMILES CC(=O)N1CCc2c(C1)c(nn2C1CCOCC1)-c1cccc2cc(ncc12)-c1ccc(nc1)C(=O)N1CC2(CC(C2)Nc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)C1

InChI Key InChIKey=ANFFPFFAJDSUIN-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50622581   

TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622581(CHEMBL5402691)
Affinity DataEC50:  0.300nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone acetyltransferase p300(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622581(CHEMBL5402691)
Affinity DataEC50:  1.10nMAssay Description:Induction of p300 degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed