BDBM50623874 CHEMBL5439595

SMILES COc1cc2nccc(Oc3ccc(NC(=O)NC4CC4)c(Cl)c3)c2cc1C1CCN(CC1)C(=O)C=C

InChI Key InChIKey=RJOWKASSFBQDER-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50623874   

TargetFibroblast growth factor receptor 4(Human)
Skyrun Pharma Co.

Curated by ChEMBL
LigandPNGBDBM50623874(CHEMBL5439595)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of FGFR4 (unknown origin) incubated for 10 mins followed by substrate addition measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetFibroblast growth factor receptor 2(Human)
Skyrun Pharma Co.

Curated by ChEMBL
LigandPNGBDBM50623874(CHEMBL5439595)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of FGFR2 (unknown origin) incubated for 10 mins followed by substrate addition measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetFibroblast growth factor receptor 4(Human)
Skyrun Pharma Co.

Curated by ChEMBL
LigandPNGBDBM50623874(CHEMBL5439595)
Affinity DataIC50: 7nMAssay Description:Inhibition of FGFR4 (unknown origin) incubated for 10 mins followed by substrate addition measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetFibroblast growth factor receptor 1(Human)
Skyrun Pharma Co.

Curated by ChEMBL
LigandPNGBDBM50623874(CHEMBL5439595)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of FGFR1 (unknown origin) incubated for 10 mins followed by substrate addition measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetFibroblast growth factor receptor 3(Human)
Skyrun Pharma Co.

Curated by ChEMBL
LigandPNGBDBM50623874(CHEMBL5439595)
Affinity DataIC50: 16nMAssay Description:Inhibition of FGFR3 (unknown origin) incubated for 10 mins followed by substrate addition measured after 60 mins by ADP-Glo luminescence assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed