BDBM50634839 CHEMBL5531958

SMILES N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN(CCCCCF)CC5)CC4)nn3)CC2)cc1Cl

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50634839   

TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634839(CHEMBL5531958)
Affinity DataIC50: 5.70nMAssay Description:Binding affinity to human androgen receptor transfected in HEK293 cell membrane co-transfected with ARC1 assessed as inhibition of [3H]-methyltrienol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
Yantai University

Curated by ChEMBL
LigandPNGBDBM50634839(CHEMBL5531958)
Affinity DataIC50: 319nMAssay Description:Antagonist activity at androgen receptor (unknown origin) transfected in HEK293T cells co-transfected with luciferase reporter gene assessed as inhib...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed