BDBM50635245 CHEMBL5549757

SMILES Cc1ccc2c(=O)c(-c3nc(-c4ccccc4C)no3)cn(CC(=O)NCCc3ccc(Cl)cc3)c2c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50635245   

TargetUbiquitin carboxyl-terminal hydrolase 10(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50635245(CHEMBL5549757)
Affinity DataKd:  5.24E+3nMAssay Description:Binding affinity to GFP tagged human USP10 assessed as dissociation constant by Microscale thermophoresis analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetUbiquitin carboxyl-terminal hydrolase 10(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50635245(CHEMBL5549757)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human USP10 deubiquitinase activity using Ubiquitin 7-amino-4-carbamoylmethylcoumarin as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed