BDBM50638324 CHEMBL2398613

SMILES CCOC(=O)[C@@H]1CS[C@@]2(C(=O)Nc3ccc(Br)cc32)N1C(=O)c1ccc(Cl)cc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50638324   

TargetPotassium channel subfamily T member 1(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50638324(CHEMBL2398613)
Affinity DataIC50: 200nMAssay Description:Inhibition of human KCNT1 (98 to 354 residues) expressed in CHO cells at +60 mV holding potential by whole-cell patch clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPotassium channel subfamily T member 1(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50638324(CHEMBL2398613)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of human KCNT1 (98 to 354 residues) expressed in CHO cells assessed as reduction in thallium fluorescent signal incubated for 15 mins foll...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed