BDBM50640862 CHEMBL4303616
SMILES CC(ONC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)Nc1ccc(Cl)cc1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50640862
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human ClpP expressed in Escherichia coli using AC-WLA-AMC as substrate measured every 5 mins for 1 hr by fluorescence based analy...More data for this Ligand-Target Pair
TargetATP-dependent Clp protease proteolytic subunit, mitochondrial(Human)
Sichuan University
Curated by ChEMBL
Sichuan University
Curated by ChEMBL
Affinity DataKd: 8.41E+3nMAssay Description:Binding affinity to human ClpP expressed in Escherichia coli assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
