BDBM50642130 CHEMBL5592453

SMILES COC(=O)c1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc2c(c1)CCN2C(=O)CN1CCOCC1)c1ccccc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50642130   

TargetPlatelet-derived growth factor receptor beta(Human)
Institute of Respiratory Health

Curated by ChEMBL
LigandPNGBDBM50642130(CHEMBL5592453)
Affinity DataIC50: 25nMAssay Description:Inhibition of PDGFRbeta (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Institute of Respiratory Health

Curated by ChEMBL
LigandPNGBDBM50642130(CHEMBL5592453)
Affinity DataIC50: 100nMAssay Description:Inhibition of glutathione S-transferase fused PDGFbetaR (unknown origin) in 3T3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Institute of Respiratory Health

Curated by ChEMBL
LigandPNGBDBM50642130(CHEMBL5592453)
Affinity DataIC50: 110nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetFibroblast growth factor receptor 1(Human)
Institute of Respiratory Health

Curated by ChEMBL
LigandPNGBDBM50642130(CHEMBL5592453)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed