BDBM50642262 CHEMBL5572993

SMILES O=c1c2nnc(C3(C4CC4)CC3)n2c2c(n1CC1CC1)CCCC2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50642262   

LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of PDE1C (unknown origin) expressed in Escherichia coli BL21 using [3H]cGMP as substrate incubated for 15 mins by liquid scintillation met...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of PDE1C (unknown origin) using [3H]-cAMP as substrate incubated for 1 hr by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of PDE1B (unknown origin) using [3H]-cGMP substrate incubated for 15 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of PDE1B (unknown origin) using [3H]-cAMP as substrate incubated for 1 hr by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 1nMAssay Description:Inhibition of PDE1A (unknown origin) using [3H]-cAMP as substrate incubated for 1 hr by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 1nMAssay Description:Inhibition of full-length recombinant human PDE1A using [3H]-cGMP as substrate incubated for 10 mins by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant full length PDE10AMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDE5A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of PDE4D (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642262(CHEMBL5572993)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PDE3A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed