BDBM50642423 CHEMBL5567321
SMILES CCn1cnc2c(NCc3ccc(-n4nc(C)cc4N)nc3)nc(N3CCCC[C@H]3CCO)nc21
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50642423
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human CDK12/Cyclin K using RNA Pol II-CTD as substrate preincubated for ~20 mins followed by 33P-ATP addition measured afte...More data for this Ligand-Target Pair
