BDBM50644322 CHEMBL5572574

SMILES CN1CCN(C(c2ccccn2)c2nnnn2Cc2ccccc2)CC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50644322   

TargetExcitatory amino acid transporter 1(Human)
Drexel University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50644322(CHEMBL5572574)
Affinity DataIC50: 1.80nMAssay Description:Negative allosteric modulation of EAAT1 (unknown origin) transfected in African green monkey COS-7 cells assessed as increase in glutamate uptake pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed