BDBM50644329 CHEMBL1393473

SMILES COc1ccc(C(c2nnnn2CCc2ccccc2)N2CCN(C)CC2)cc1OC

InChI Key InChIKey=VFMUGBFABSUSKZ-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50644329   

TargetExcitatory amino acid transporter 3(Human)
Drexel University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50644329(CHEMBL1393473)
Affinity DataEC50:  132nMAssay Description:Positive allosteric modulation of EAAT3 (unknown origin) transfected in African green monkey COS-7 cells assessed as increase in glutamate uptake pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetExcitatory amino acid transporter 1(Human)
Drexel University College of Medicine

Curated by ChEMBL
LigandPNGBDBM50644329(CHEMBL1393473)
Affinity DataEC50:  132nMAssay Description:Positive allosteric modulation of EAAT1 (unknown origin) transfected in African green monkey COS-7 cells assessed as increase in glutamate uptake pre...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed