BDBM50644632 CHEMBL5564481

SMILES CC(=O)c1c[nH]c2cc3cnccc3cc12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50644632   

TargetSerine/threonine-protein kinase haspin(Human)
Universite Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50644632(CHEMBL5564481)
Affinity DataIC50: 157nMAssay Description:Inhibition of recombinant human Haspin kinase domain (470 to 798 residues) expressed in bacteria using histone H3 (1 to 21) peptide as substrate incu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Universite Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50644632(CHEMBL5564481)
Affinity DataIC50: 265nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate incubated for 30 mins in presence of ATP by ADP-Glo kinase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Universite Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50644632(CHEMBL5564481)
Affinity DataIC50: 860nMAssay Description:Inhibition of recombinant rat DYRK1A kinase domain (1 to 499 residues) expressed in bacteria using KKISGRLSPIMTEQ as substrate incubated for 30 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed