BDBM50645052 CHEMBL5564691

SMILES COc1ccc(C2COc3cc(OCc4c(C)cc(C)cc4C)ccc3C2=O)cc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50645052   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at capsaicin activated human TRPV1 expressed in HEK293 cells incubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 9.71E+3nMAssay Description:Inhibition of human TRPV1 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TRPA1 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TRPV4 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 3(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TRPV3 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed