BDBM50645344 CHEMBL5571203

SMILES O=C(O)[C@H]1CCCN(c2ncnc3ccc(-c4c[nH]c5ncccc45)cc23)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50645344   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50645344(CHEMBL5571203)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of DYRK1A (unknown origin) preincubated with enzyme for 10 mins followed by substrate and ATP addition measured after 60 mins by ADP-Glo r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed