BDBM50646127 CHEMBL5593461

SMILES O=C(O)CCCc1cnnn1[C@H]1CN[C@H](C(=O)O)[C@H]1CC(=O)O

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50646127   

TargetGlutamate receptor ionotropic, kainate 5(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646127(CHEMBL5593461)
Affinity DataKi:  483nMAssay Description:Displacement of [3H]-kainate from mouse GluK5 expressed in Sf9 cell membrane incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646127(CHEMBL5593461)
Affinity DataKi:  6.10E+3nMAssay Description:Displacement of [3H]-KA from rat GluK3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646127(CHEMBL5593461)
Affinity DataKi:  7.79E+3nMAssay Description:Displacement of [3H]-KA from rat GluK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlutamate receptor ionotropic, kainate 1(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646127(CHEMBL5593461)
Affinity DataKi:  1.08E+4nMAssay Description:Displacement of [3H]-NF608 from rat GluK1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed