BDBM50646128 CHEMBL5594100

SMILES O=C(O)C[C@@H]1[C@@H](C(=O)O)NC[C@@H]1n1nncc1-c1ccccn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50646128   

TargetGlutamate receptor ionotropic, kainate 5(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646128(CHEMBL5594100)
Affinity DataKi:  258nMAssay Description:Displacement of [3H]-kainate from mouse GluK5 expressed in Sf9 cell membrane incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlutamate receptor ionotropic, kainate 3(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646128(CHEMBL5594100)
Affinity DataKi:  3.75E+3nMAssay Description:Displacement of [3H]-KA from rat GluK3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646128(CHEMBL5594100)
Affinity DataKi:  7.76E+3nMAssay Description:Displacement of [3H]-KA from rat GluK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlutamate receptor ionotropic, kainate 1(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50646128(CHEMBL5594100)
Affinity DataKi:  1.15E+4nMAssay Description:Displacement of [3H]-NF608 from rat GluK1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed