BDBM50646762 CHEMBL5592836

SMILES CC1(NC(=O)c2cn3cc(Oc4ncc(F)cc4OCC(F)(F)F)ccc3n2)CCS(=O)(=O)CC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50646762   

TargetDiacylglycerol O-acyltransferase 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50646762(CHEMBL5592836)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human DGAT2 extracted from baculovirus infected Sf9 cell membrane using 13C-oleoyl-CoA as substrate by measuring [13C]18-triolein produ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDiacylglycerol O-acyltransferase 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50646762(CHEMBL5592836)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human DGAT2 expressed in expressed in baculovirus infected Sf9 insect cells by immunoblotting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed