BDBM50646847 CHEMBL5594658

SMILES C[C@H](Oc1ccc2c(c1)OCc1ccc(-c3ncnn3C)cc1-2)C(N)=O

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50646847   

LigandPNGBDBM50646847(CHEMBL5594658)
Affinity DataIC50: 17nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo reagent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50646847(CHEMBL5594658)
Affinity DataIC50: 933nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo reagent assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50646847(CHEMBL5594658)
Affinity DataIC50: 4.97E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo reagent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50646847(CHEMBL5594658)
Affinity DataIC50: 5.07E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo reagent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed