BDBM50647389 CHEMBL5590573

SMILES [2H]C([2H])([2H])OC(c1ccc(F)cc1C(F)(F)F)c1cnc2n1CCN(c1cn[nH]c(=O)c1Cl)C2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50647389   

TargetShort transient receptor potential channel 5(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50647389(CHEMBL5590573)
Affinity DataIC50: 19nMAssay Description:Inhibition of TRPC5 (unknown origin) expressed in HEK293 cells assessed as reduction in englerin A stimulated Ca2+ influx by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed