BDBM50647407 CHEMBL5589721

SMILES COC(c1ccc(F)cc1Cl)c1c(C(F)(F)F)nc2n1CCN(c1cn[nH]c(=O)c1Cl)C2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50647407   

TargetShort transient receptor potential channel 5(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50647407(CHEMBL5589721)
Affinity DataIC50: 249nMAssay Description:Inhibition of TRPC5 (unknown origin) expressed in HEK293 cells assessed as reduction in englerin A stimulated Ca2+ influx by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed