BDBM50648670 CHEMBL5612930

SMILES Cc1ncncc1Nc1ccc2c(c1)CCC1=C3C[C@@H](O)C[C@]3(C)CC[C@]12Cc1ccccc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50648670   

TargetProgesterone receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human PGR transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene assessed as inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at full length glucocorticoid receptor (unknown origin) assessed as inhibition of Fluormone GS Red binding to receptor incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 131nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in HEK293 cells cotransfected with genetic response element-luciferase reporter gene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50648670(CHEMBL5612930)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human androgen receptor transfected in African green monkey CV-1 cells cotransfected with genetic response element-luciferase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed