BDBM50649419 CHEMBL5618375

SMILES C/C(=C\Cc1cccc2c1OC(c1ccc(Br)c3ccccc13)CC2=O)C(=O)O

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50649419   

TargetSolute carrier family 22 member 12(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50649419(CHEMBL5618375)
Affinity DataIC50: 160nMAssay Description:Inhibition of human URAT1 transfected in HEK293 cells by measuring 14C-uric acid uptake preincubated for 30 mins followed by 14--uric acid addition a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 9(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50649419(CHEMBL5618375)
Affinity DataIC50: 4.47E+3nMAssay Description:Inhibition of GLUT9 (unknown origin) overexpressed in uric acid-induced HEK293 cells by patch clamp analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed