BDBM50650244 CHEMBL5624805

SMILES O=C(Nc1nccs1)c1ccc(NC(=O)[C@@H]2C[C@H]2c2ccccc2)cc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50650244   

TargetSodium channel protein type 3 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 990nMAssay Description:Inhibition of human Nav1.3 expressed in CHO cells under inactivated state by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium channel protein type 3 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human Nav1.3 expressed in CHO cells under resting state by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.7 expressed in CHO cells under inactivated state by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 expressed in CHO cells under resting state by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.7 expressed in CHO cells under resting state by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 expressed in CHO cells under phasic pulse 1 by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 expressed in CHO cells under tonic pulse 1 by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50650244(CHEMBL5624805)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 expressed in CHO cells under inactivated state by automated patch clamp electrophysiology analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed