BDBM50651356 CHEMBL5633177

SMILES CN(C)CCN1CCC(NC(=O)c2ccc3c(Nc4ccc(CN)cc4)ncnc3c2)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50651356   

TargetProtein arginine N-methyltransferase 1(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651356(CHEMBL5633177)
Affinity DataIC50: 1.50E+4nMAssay Description:Displacement of 3H-SAM from PRMT1 (unknown origin) using biotinylated-histone H4 peptide as substrate incubated for 45 mins by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase SUV39H1(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651356(CHEMBL5633177)
Affinity DataIC50: 1.60E+4nMAssay Description:Displacement of 3H-SAM from SUV39H1 (unknown origin) using biotinylated-histone H3 peptide as substrate incubated for 45 mins by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed