BDBM50651357 CHEMBL5633967

SMILES CNCCN1CCC(NC(=O)c2ccc3c(Nc4ccc(CN)cc4)ncnc3c2)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50651357   

TargetProtein arginine N-methyltransferase 1(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651357(CHEMBL5633967)
Affinity DataIC50: 2.43E+3nMAssay Description:Displacement of 3H-SAM from PRMT1 (unknown origin) using biotinylated-histone H4 peptide as substrate incubated for 45 mins by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651357(CHEMBL5633967)
Affinity DataIC50: 8.00E+4nMAssay Description:Displacement of 3H-SAM from human PRMT4 in presence of substrate by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651357(CHEMBL5633967)
Affinity DataIC50: 7.03E+5nMAssay Description:Displacement of 3H-SAM from human PRMT6 in presence of substrate by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651357(CHEMBL5633967)
Affinity DataIC50: 2.43E+6nMAssay Description:Displacement of 3H-SAM from human PRMT8 in presence of substrate by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651357(CHEMBL5633967)
Affinity DataIC50: 2.43E+6nMAssay Description:Displacement of 3H-SAM from human PRMT1 in presence of substrate by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
CSIR-Indian Institute of Chemical Biology (IICB)

Curated by ChEMBL
LigandPNGBDBM50651357(CHEMBL5633967)
Affinity DataIC50: 3.12E+6nMAssay Description:Displacement of 3H-SAM from human PRMT3 in presence of substrate by SPA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed