BDBM50652735 CHEMBL1254460

SMILES O=C1/C(=C/c2ccccc2Cl)CNC/C1=C\c1ccccc1Cl

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50652735   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50652735(CHEMBL1254460)
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant DYRK2 using KKISGRLSPIMTEQ as substrate incubated for 60 mins in the presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50652735(CHEMBL1254460)
Affinity DataKd:  4.70E+3nMAssay Description:Binding affinity to DYRK2 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed