BDBM50652775 CHEMBL4303308
SMILES O=C(O)CCNc1cc(N2CCc3ccccc3CC2)nc(-c2cccnc2)n1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 18 hits for monomerid = 50652775
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM3B (842 to 1761 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM4A (1 to 350 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM4B (2 to 500 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM4C (1 to 349 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM3A (2 to 1322 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of KDM6A (919 to 1401 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of epitope-tagged KDM6B (1026 to 1682 residues)(unknown origin) transfected in human U2OS cells using H3K27me2 peptide as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PHF8 (1 to 1024 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of KDM5A (1 to 1090 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibition of KDM5B (1 to 809 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition of KDM6B (1043 to 1643 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Inhibition of KDM5C (2 to 1560 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30nMAssay Description:Inhibition of KDM2B (1 to 650 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition of human JmjD2c using H3K27(me3) as substrate preincubated for 10 mins followed by substrate addition and measured after 7 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JmjD2a using H3K27(me3) as substrate preincubated for 10 mins followed by substrate addition and measured after 7 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JmjD2d using H3K27(me3) as substrate preincubated for 10 mins followed by substrate addition and measured after 7 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JmjD2e using H3K27(me3) as substrate preincubated for 10 mins followed by substrate addition and measured after 7 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His6/Flag-tagged TEV-protease cleavage site fused JMJD3 1637-1675 deletion mutant (1141 to 1682 residues) ...More data for this Ligand-Target Pair