BDBM50652834 CHEMBL5661924
SMILES Cc1nn(CCc2ccc(F)cc2)c(C)c1NC(=O)c1cc(C(F)(F)F)nc2ccc(Br)cc12
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50652834
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Bayer AG
Curated by ChEMBL
Bayer AG
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of human GLUT1 expressed in human DLD-1 cells assessed as reduction in glucose uptake by measuring decrease in ATP production incubated fo...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 4(Human)
Bayer AG
Curated by ChEMBL
Bayer AG
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of human GLUT4 expressed in CHO cells assessed as reduction in glucose uptake by measuring decrease in ATP production preincubated for 20 ...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 3(Human)
Bayer AG
Curated by ChEMBL
Bayer AG
Curated by ChEMBL
Affinity DataIC50: 2.39E+3nMAssay Description:Inhibition of human GLUT3 expressed in human GLUT1-/- DLD-1 cells assessed as reduction in glucose uptake by measuring decrease in ATP production inc...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 2(Human)
Bayer AG
Curated by ChEMBL
Bayer AG
Curated by ChEMBL
Affinity DataIC50: 5.63E+3nMAssay Description:Inhibition of human GLUT2 expressed in CHO cells assessed as reduction in fructose uptake by measuring decrease in ATP production incubated for 15 mi...More data for this Ligand-Target Pair