BDBM50653002 CHEMBL1643976

SMILES C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(C)CC4)cc3)ncc2Cl)c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50653002   

LigandPNGBDBM50653002(CHEMBL1643976)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of TEL fused BMX (unknown origin) transformed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50653002(CHEMBL1643976)
Affinity DataIC50: 20nMAssay Description:Inhibition of TEL fused BLK (unknown origin) transformed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50653002(CHEMBL1643976)
Affinity DataIC50: 35nMAssay Description:Inhibition of TEL fused JAK3 (unknown origin) transformed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50653002(CHEMBL1643976)
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of wildtype EGFR (unknown origin) transformed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50653002(CHEMBL1643976)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of TEL fused JAK2 (unknown origin) transformed in mouse BaF3 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed